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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T62797 | A2A receptor antagonist 3 | ||
A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM). | |||
T6552 | Istradefylline | KW-6002 | Adenosine Receptor |
Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in trials studying the treatment and basic science of Drug Ab... | |||
T25841 | MSX-3 | MSX 3 | |
MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2. | |||
T69566 | MSX-3 free acid | ||
MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2. | |||
T62611 | Adenosine receptor antagonist 2 | ||
Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects. | |||
T72626 | A2AR-antagonist-1 | Adenosine Receptor | |
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability in mouse liver microsomes (t1/2 = 86.1 min). Additionally,... |